OpenSourceMalaria:Compound Series: Difference between revisions

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A summary of progress in the OSM project may be found in the [[OpenSourceMalaria:Story_so_far|Story so Far]]. The pages below include the technical detail of the individual series examined and are written for scientific contributors.
A summary of progress in the OSM project may be found in the [[OpenSourceMalaria:Story_so_far|Story so Far]]. The pages below include the technical detail of the individual series examined and are written for scientific contributors.


[[OpenSourceMalaria:GSK_Arylpyrrole_Series |'''Series 1: GSK Arylpyrroles''']] (being written up)
[[OpenSourceMalaria:GSK_Arylpyrrole_Series |'''Series 1: GSK Arylpyrroles''']] (Paper has been released: http://pubs.acs.org/doi/full/10.1021/acscentsci.6b00086)


[[OpenSourceMalaria:GSK_Triazolourea_Singleton |'''Series 2: GSK Triazoloureas''']] (parked)
[[OpenSourceMalaria:GSK_Triazolourea_Singleton |'''Series 2: GSK Triazoloureas''']] (parked)


[[OpenSourceMalaria:GSK_Amino-thienopyrimidine_Series |'''Series 3: GSK Thienopyrimidines''']] (final compounds being made)
[[OpenSourceMalaria:GSK_Amino-thienopyrimidine_Series |'''Series 3: GSK Thienopyrimidines''']] (work is resuming)


[[OpenSourceMalaria:Triazolopyrazine_(TP)_Series |'''Series 4: Triazolopyrazines (TPs)''']] (currently most active)
[[OpenSourceMalaria:Triazolopyrazine_(TP)_Series |'''Series 4: Triazolopyrazines (TP series)''']] (current priority)
 
[[OpenSourceMalaria:Triazolopyrazine_Series Mechanism of Action |'''Series 4: Mechanism of Action''']]


[[OpenSourceMalaria:Synthesis Branches |'''Synthetic Branches''']]
[[OpenSourceMalaria:Synthesis Branches |'''Synthetic Branches''']]

Latest revision as of 11:24, 27 May 2017

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A summary of progress in the OSM project may be found in the Story so Far. The pages below include the technical detail of the individual series examined and are written for scientific contributors.

Series 1: GSK Arylpyrroles (Paper has been released: http://pubs.acs.org/doi/full/10.1021/acscentsci.6b00086)

Series 2: GSK Triazoloureas (parked)

Series 3: GSK Thienopyrimidines (work is resuming)

Series 4: Triazolopyrazines (TP series) (current priority)

Series 4: Mechanism of Action

Synthetic Branches

Obtaining Compounds for OSM

Repurposing

Other Possible GSK Series

Other Possible Series and Targets

Epigenetic Regulation of Lifecycle